26 Sep, 2025 Publications

Enantioselective Synthesis of a 2,3-Benzodiazepine Intermediate of BET Inhibitor BAY 1238097 via Catalytic Asymmetric Hydrogenation


Verzijl, Gerard; Hassfeld Jorma; de Vries Andre; Lefort Laurent


Enantioselective Synthesis of a 2,3-Benzodiazepine Intermediate of BET Inhibitor BAY 1238097 via Catalytic Asymmetric Hydrogenation.


Org. Process Res. Dev. (2020), 24, 2, 255–260. DOI/10.1021/acs.oprd.9b00519