Enantioselective Synthesis of a 2,3-Benzodiazepine Intermediate of BET Inhibitor BAY 1238097 via Catalytic Asymmetric Hydrogenation

Verzijl, Gerard; Hassfeld Jorma; de Vries Andre; Lefort Laurent

Enantioselective Synthesis of a 2,3-Benzodiazepine Intermediate of BET Inhibitor BAY 1238097 via Catalytic Asymmetric Hydrogenation.

Org. Process Res. Dev. (2020), 24, 2, 255–260.
DOI/10.1021/acs.oprd.9b00519